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Target
Cathepsin G
Ligand
BDBM33426
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM33426
Synonyms:
(5-Amino-3-p-tolyl-[1,2,4]triazol-1-yl)-(3,4-dimethoxy-phenyl)-methanone | MLS000076095 | SMR000013731 | [5-amino-3-(4-methylphenyl)-1,2,4-triazol-1-yl]-(3,4-dimethoxyphenyl)methanone | [5-amino-3-(p-tolyl)-1,2,4-triazol-1-yl]-(3,4-dimethoxyphenyl)methanone | [5-azanyl-3-(4-methylphenyl)-1,2,4-triazol-1-yl]-(3,4-dimethoxyphenyl)methanone | cid_654458
Type:
Small organic molecule
Emp. Form.:
C18H18N4O3
Mol. Mass.:
338.3605
SMILES:
COc1ccc(cc1OC)C(=O)n1nc(nc1N)-c1ccc(C)cc1
Structure:
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