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Target
Cathepsin G
Ligand
BDBM41389
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41389
Synonyms:
3-(morpholin-4-ylcarbonyl)-4,5-dihydronaphtho[2,1-d]isoxazole | 4,5-dihydrobenz[g]indoxazen-3-yl(morpholino)methanone | 4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl(4-morpholinyl)methanone | 4,5-dihydrobenzo[g][1,2]benzoxazol-3-yl(morpholin-4-yl)methanone | MLS000087428 | SMR000023651 | cid_3236015
Type:
Small organic molecule
Emp. Form.:
C16H16N2O3
Mol. Mass.:
284.3098
SMILES:
O=C(N1CCOCC1)c1noc-2c1CCc1ccccc-21
Structure:
Search PDB for entries with ligand similarity: