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Target
Cathepsin G
Ligand
BDBM41404
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
11127.9±551.536 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41404
Synonyms:
MLS000087096 | N-(4-chlorobenzyl)-5-(2-methoxyphenyl)isoxazole-3-carboxamide | N-[(4-chlorophenyl)methyl]-5-(2-methoxyphenyl)-1,2-oxazole-3-carboxamide | N-[(4-chlorophenyl)methyl]-5-(2-methoxyphenyl)-3-isoxazolecarboxamide | SMR000023319 | cid_3241352
Type:
Small organic molecule
Emp. Form.:
C18H15ClN2O3
Mol. Mass.:
342.776
SMILES:
COc1ccccc1-c1cc(no1)C(=O)NCc1ccc(Cl)cc1
Structure:
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