Reaction Details Report a problem with these data
Target
Cathepsin G
Ligand
BDBM41409
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
13294.6±1247.47 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41409
Synonyms:
5-(2-methoxyphenyl)-N-(phenylmethyl)-1,2-oxazole-3-carboxamide | 5-(2-methoxyphenyl)-N-(phenylmethyl)-3-isoxazolecarboxamide | MLS000087092 | N-benzyl-5-(2-methoxyphenyl)-1,2-oxazole-3-carboxamide | N-benzyl-5-(2-methoxyphenyl)isoxazole-3-carboxamide | SMR000023315 | cid_3243790
Type:
Small organic molecule
Emp. Form.:
C18H16N2O3
Mol. Mass.:
308.3312
SMILES:
COc1ccccc1-c1cc(no1)C(=O)NCc1ccccc1
Structure:
Search PDB for entries with ligand similarity: