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Target
Cathepsin G
Ligand
BDBM32787
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
9801.24±600.84 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM32787
Synonyms:
1-[2-(ethylthio)benzoyl]-1H-1,2,3-benzotriazole | 1-benzotriazolyl-[2-(ethylthio)phenyl]methanone | MLS000050138 | SMR000077231 | benzotriazol-1-yl-(2-ethylsulfanylphenyl)methanone | benzotriazol-1-yl-[2-(ethylthio)phenyl]methanone | cid_2212050
Type:
Small organic molecule
Emp. Form.:
C15H13N3OS
Mol. Mass.:
283.348
SMILES:
CCSc1ccccc1C(=O)n1nnc2ccccc12
Structure:
Search PDB for entries with ligand similarity: