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Target
Cathepsin G
Ligand
BDBM41414
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
4656.35±241.657 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41414
Synonyms:
5-[(3-methyl-2-thienyl)methylene][1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one | 5-[(3-methyl-2-thienyl)methylene]thiazolo[3,2-b][1,2,4]triazol-6-one | 5-[(3-methyl-2-thiophenyl)methylidene]-6-thiazolo[3,2-b][1,2,4]triazolone | 5-[(3-methylthiophen-2-yl)methylidene]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one | MLS000088270 | SMR000072513 | cid_3246790
Type:
Small organic molecule
Emp. Form.:
C10H7N3OS2
Mol. Mass.:
249.312
SMILES:
Cc1ccsc1C=c1sc2ncnn2c1=O
Structure:
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