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Target
Cathepsin G
Ligand
BDBM40904
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
41519±563.3 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM40904
Synonyms:
(3-bromanyl-4-methoxy-phenyl)-(3-methylpyrazol-1-yl)methanone | (3-bromo-4-methoxy-phenyl)-(3-methylpyrazol-1-yl)methanone | (3-bromo-4-methoxyphenyl)-(3-methyl-1-pyrazolyl)methanone | (3-bromo-4-methoxyphenyl)-(3-methylpyrazol-1-yl)methanone | 1-(3-bromo-4-methoxybenzoyl)-3-methyl-1H-pyrazole | MLS000063131 | SMR000074342 | cid_899202
Type:
Small organic molecule
Emp. Form.:
C12H11BrN2O2
Mol. Mass.:
295.132
SMILES:
COc1ccc(cc1Br)C(=O)n1ccc(C)n1
Structure:
Search PDB for entries with ligand similarity: