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Target
Cathepsin G
Ligand
BDBM33609
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
4509.63±449.07 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM33609
Synonyms:
(5-azanyl-3-morpholin-4-ylcarbonyl-1,2,4-triazol-1-yl)-(4-chlorophenyl)methanone | MLS000115334 | SMR000092476 | [5-amino-3-(morpholine-4-carbonyl)-1,2,4-triazol-1-yl]-(4-chlorophenyl)methanone | [5-amino-3-[4-morpholinyl(oxo)methyl]-1,2,4-triazol-1-yl]-(4-chlorophenyl)methanone | cid_3586649
Type:
Small organic molecule
Emp. Form.:
C14H14ClN5O3
Mol. Mass.:
335.746
SMILES:
Nc1nc(nn1C(=O)c1ccc(Cl)cc1)C(=O)N1CCOCC1
Structure:
Search PDB for entries with ligand similarity: