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Target
Cathepsin G
Ligand
BDBM41419
Substrate
n/a
Meas. Tech.
Cathepsin G dose-response confirmation
IC50
4254.8±150.149 nM
Citation
 PubChem, PC Cathepsin G dose-response confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Cathepsin G
Synonyms:
CATG_HUMAN | CG | CTSG
Type:
PROTEIN
Mol. Mass.:
28860.08
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1469016
Residue:
255
Sequence:
MQPLLLLLAFLLPTGAEAGEIIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSFKLLDQMETPL
  
Inhibitor
Name:
BDBM41419
Synonyms:
MLS000116422 | N-(5-methyl-1,2-oxazol-3-yl)-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamide | N-(5-methyl-3-isoxazolyl)-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamide | N-(5-methylisoxazol-3-yl)-4,5-dihydrobenz[g]indoxazene-3-carboxamide | SMR000093399 | cid_5309278
Type:
Small organic molecule
Emp. Form.:
C16H13N3O3
Mol. Mass.:
295.2927
SMILES:
Cc1cc(NC(=O)c2noc-3c2CCc2ccccc-32)no1
Structure:
Search PDB for entries with ligand similarity: