Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43672
Substrate
n/a
Meas. Tech.
Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43672
Synonyms:
2-ethoxy-N-(6-ethoxy-1,3-benzothiazol-2-yl)acetamide | 2-ethoxy-N-(6-ethoxy-1,3-benzothiazol-2-yl)ethanamide | MLS000064361 | SMR000076590 | cid_2206392
Type:
Small organic molecule
Emp. Form.:
C13H16N2O3S
Mol. Mass.:
280.343
SMILES:
CCOCC(=O)Nc1nc2ccc(OCC)cc2s1
Structure:
Search PDB for entries with ligand similarity: