Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43707
Substrate
n/a
Meas. Tech.
Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43707
Synonyms:
2-(2-phenyl-1,3-benzothiazol-5-yl)acetamide | 2-(2-phenyl-1,3-benzothiazol-5-yl)ethanamide | MLS000391716 | SMR000260751 | cid_726461
Type:
Small organic molecule
Emp. Form.:
C15H12N2OS
Mol. Mass.:
268.334
SMILES:
NC(=O)Cc1ccc2sc(nc2c1)-c1ccccc1
Structure:
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