Reaction Details Report a problem with these data
Target
Protein Rev [8-24]
Ligand
BDBM44538
Substrate
n/a
Meas. Tech.
Dose response biochemical assay to identify inhibitors of the HIV Rev - RRE RNA interaction (disruption of protein-RNA interaction)
IC50
>79370±n/a nM
Citation
 PubChem, PC Dose response biochemical assay to identify inhibitors of the HIV Rev - RRE RNA interaction (disruption of protein-RNA interaction) PubChem Bioassay (2007)[AID] 
Target
Name:
Protein Rev [8-24]
Synonyms:
Chain B, Rna Aptamer Complexed With Hiv-1 Rev Peptide, Nmr, 7 Structures | REV_HV1W2 | rev
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2446.81
Organism:
Human immunodeficiency virus 1
Description:
gi_253722402
Residue:
17
Sequence:
TRQARRNRRRRWRERQR
  
Inhibitor
Name:
BDBM44538
Synonyms:
4-Amino-1-phenothiazin-10-yl-butan-1-one | 4-amino-1-(10-phenothiazinyl)-1-butanone;hydrochloride | 4-amino-1-phenothiazin-10-yl-butan-1-one;hydrochloride | 4-amino-1-phenothiazin-10-ylbutan-1-one;hydrochloride | 4-azanyl-1-phenothiazin-10-yl-butan-1-one;hydrochloride | MLS000120403 | SMR000102020 | cid_6603292
Type:
Small organic molecule
Emp. Form.:
C16H16N2OS
Mol. Mass.:
284.376
SMILES:
NCCCC(=O)N1c2ccccc2Sc2ccccc12
Structure:
Search PDB for entries with ligand similarity: