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Target
Sphingosine 1-phosphate receptor 2
Ligand
BDBM41679
Substrate
n/a
Meas. Tech.
Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA
EC50
>50000±n/a nM
Citation
 PubChem, PC Counter screen for S1P2 Agonists: Dose Response High Throughput Cell-Based Screen to Identify Activators of CRE-BLA PubChem Bioassay (2007)[AID] 
Target
Name:
Sphingosine 1-phosphate receptor 2
Synonyms:
EDG5 | S1P2 | S1PR2 | S1PR2_HUMAN | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor Edg-5 | Sphingosine-1-phosphate receptor 2 | ndothelial differentiation G-protein coupled receptor 5
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38883.16
Organism:
Homo sapiens (Human)
Description:
Membranes isolated from S1P2-transfected CHO cells were used in ligand binding assay.
Residue:
353
Sequence:
MGSLYSEYLNPNKVQEHYNYTKETLETQETTSRQVASAFIVILCCAIVVENLLVLIAVARNSKFHSAMYLFLGNLAASDLLAGVAFVANTLLSGSVTLRLTPVQWFAREGSAFITLSASVFSLLAIAIERHVAIAKVKLYGSDKSCRMLLLIGASWLISLVLGGLPILGWNCLGHLEACSTVLPLYAKHYVLCVVTIFSIILLAIVALYVRIYCVVRSSHADMAAPQTLALLKTVTIVLGVFIVCWLPAFSILLLDYACPVHSCPILYKAHYFFAVSTLNSLLNPVIYTWRSRDLRREVLRPLQCWRPGVGVQGRRRGGTPGHHLLPLRSSSSLERGMHMPTSPTFLEGNTVV
  
Inhibitor
Name:
BDBM41679
Synonyms:
6-Methoxy-naphthalene-2-sulfonic acid (3-morpholin-4-yl-propyl)-amide | 6-methoxy-N-(3-morpholin-4-ylpropyl)naphthalene-2-sulfonamide | 6-methoxy-N-(3-morpholinopropyl)naphthalene-2-sulfonamide | 6-methoxy-N-[3-(4-morpholinyl)propyl]-2-naphthalenesulfonamide | MLS000026958 | SMR000122898 | cid_2280707
Type:
Small organic molecule
Emp. Form.:
C18H24N2O4S
Mol. Mass.:
364.459
SMILES:
COc1ccc2cc(ccc2c1)S(=O)(=O)NCCCN1CCOCC1
Structure:
Search PDB for entries with ligand similarity: