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Target
Regulator of G-protein signaling 8
Ligand
BDBM47768
Substrate
n/a
Meas. Tech.
Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 8
Synonyms:
RGS8 | RGS8_HUMAN | Regulator of G-protein signaling 8 (RGS8)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
20925.80
Organism:
Homo sapiens (Human)
Description:
gi_74355113
Residue:
180
Sequence:
MAALLMPRRNKGMRTRLGCLSHKSDSCSDFTAILPDKPNRALKRLSTEEATRWADSFDVLLSHKYGVAAFRAFLKTEFSEENLEFWLACEEFKKTRSTAKLVSKAHRIFEEFVDVQAPREVNIDFQTREATRKNLQEPSLTCFDQAQGKVHSLMEKDSYPRFLRSKMYLDLLSQSQRRLS
  
Inhibitor
Name:
BDBM47768
Synonyms:
MLS000681208 | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxy-benzamide | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxybenzamide | SMR000269463 | cid_1562455
Type:
Small organic molecule
Emp. Form.:
C18H21NO3
Mol. Mass.:
299.3642
SMILES:
COc1cccc(c1)C(=O)NCCOc1cc(C)cc(C)c1
Structure:
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