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Target
Regulator of G-protein signaling 19
Ligand
BDBM47727
Substrate
n/a
Meas. Tech.
Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 19
Synonyms:
G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24631.38
Organism:
Homo sapiens (Human)
Description:
gi_86990435
Residue:
217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFWLACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDAQLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
  
Inhibitor
Name:
BDBM47727
Synonyms:
3-Methyl-benzoic acid N'-(tetrahydro-furan-2-carbonyl)-hydrazide | MLS000555698 | N'-(3-methylbenzoyl)oxolane-2-carbohydrazide | N'-(3-methylphenyl)carbonyloxolane-2-carbohydrazide | N'-[(3-methylphenyl)-oxomethyl]-2-oxolanecarbohydrazide | N'-m-toluoyltetrahydrofuran-2-carbohydrazide | SMR000176702 | cid_3128422
Type:
Small organic molecule
Emp. Form.:
C13H16N2O3
Mol. Mass.:
248.2777
SMILES:
Cc1cccc(c1)C(=O)NNC(=O)C1CCCO1
Structure:
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