Target
Regulator of G-protein signaling 19
Ligand
BDBM47768
Substrate
n/a
Meas. Tech.
Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 19
Synonyms:
G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24631.38
Organism:
Homo sapiens (Human)
Description:
gi_86990435
Residue:
217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFWLACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDAQLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
  
Inhibitor
Name:
BDBM47768
Synonyms:
MLS000681208 | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxy-benzamide | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxybenzamide | SMR000269463 | cid_1562455
Type:
Small organic molecule
Emp. Form.:
C18H21NO3
Mol. Mass.:
299.3642
SMILES:
COc1cccc(c1)C(=O)NCCOc1cc(C)cc(C)c1
Structure:
Search PDB for entries with ligand similarity: