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Target
Regulator of G-protein signaling 19
Ligand
BDBM47800
Substrate
n/a
Meas. Tech.
Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 19
Synonyms:
G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24631.38
Organism:
Homo sapiens (Human)
Description:
gi_86990435
Residue:
217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFWLACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDAQLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
  
Inhibitor
Name:
BDBM47800
Synonyms:
MLS000736409 | N'-[(E)-(2-fluorophenyl)methylidene]benzenesulfonohydrazide | N-[(2-fluorobenzylidene)amino]benzenesulfonamide | N-[(2-fluorophenyl)methylideneamino]benzenesulfonamide | SMR000338359 | cid_2172475
Type:
Small organic molecule
Emp. Form.:
C13H11FN2O2S
Mol. Mass.:
278.302
SMILES:
Fc1ccccc1C=NNS(=O)(=O)c1ccccc1 |w:8.9|
Structure:
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