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Target
Regulator of G-protein signaling 19
Ligand
BDBM47810
Substrate
n/a
Meas. Tech.
Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 19
Synonyms:
G protein signalling regulator 19 | GAIP | GNAI3IP | RGS19 | RGS19_HUMAN | Regulator of G-protein signaling 19 (RGS19)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24631.38
Organism:
Homo sapiens (Human)
Description:
gi_86990435
Residue:
217
Sequence:
MPTPHEAEKQITGPEEADRPPSMSSHDTASPAAPSRNPCCLCWCCCCSCSWNQERRRAWQASRESKLQPLPSCEVCATPSPEEVQSWAQSFDKLMHSPAGRSVFRAFLRTEYSEENMLFWLACEELKAEANQHVVDEKARLIYEDYVSILSPKEVSLDSRVREGINKKMQEPSAHTFDDAQLQIYTLMHRDSYPRFLSSPTYRALLLQGPSQSSSEA
  
Inhibitor
Name:
BDBM47810
Synonyms:
2-(pyridin-4-ylcarbonylamino)ethyl N-(3,4-dichlorophenyl)carbamate | 2-(pyridine-4-carbonylamino)ethyl N-(3,4-dichlorophenyl)carbamate | MLS001034017 | N-(3,4-dichlorophenyl)carbamic acid 2-[[oxo(pyridin-4-yl)methyl]amino]ethyl ester | N-(3,4-dichlorophenyl)carbamic acid 2-isonicotinamidoethyl ester | SMR000385849 | cid_2121675
Type:
Small organic molecule
Emp. Form.:
C15H13Cl2N3O3
Mol. Mass.:
354.188
SMILES:
Clc1ccc(NC(=O)OCCNC(=O)c2ccncc2)cc1Cl
Structure:
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