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Target
Regulator of G-protein signaling 16
Ligand
BDBM47720
Substrate
n/a
Meas. Tech.
Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 16
Synonyms:
RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22748.87
Organism:
Homo sapiens (Human)
Description:
gi_156416009
Residue:
202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVLGWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEEFICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDLAAQASAASATLSSCSLDEPSHT
  
Inhibitor
Name:
BDBM47720
Synonyms:
2-N,2-N-diethyl-4-N,4-N-diphenyl-1,3,5-triazine-2,4,6-triamine | MLS000522302 | N2,N2-diethyl-N4,N4-diphenyl-1,3,5-triazine-2,4,6-triamine | SMR000127570 | [4-amino-6-(diethylamino)-s-triazin-2-yl]-diphenyl-amine | cid_712290
Type:
Small organic molecule
Emp. Form.:
C19H22N6
Mol. Mass.:
334.4182
SMILES:
CCN(CC)c1nc(N)nc(n1)N(c1ccccc1)c1ccccc1
Structure:
Search PDB for entries with ligand similarity: