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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM39080
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
770±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM39080
Synonyms:
4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butanoic acid | 4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]butyric acid | MLS000042181 | SMR000048679 | cid_667316
Type:
Small organic molecule
Emp. Form.:
C13H14N2O4
Mol. Mass.:
262.2613
SMILES:
COc1ccc(cc1)-c1noc(CCCC(O)=O)n1
Structure:
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