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Target
D(1B) dopamine receptor
Ligand
BDBM48967
Substrate
n/a
Meas. Tech.
Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen
EC50
0.0402±n/a nM
Citation
 PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Counterscreen PubChem Bioassay (2007)[AID] 
Target
Name:
D(1B) dopamine receptor
Synonyms:
D(5) dopamine receptor | D1beta dopamine receptor | DOPAMINE D5 | DRD1B | DRD1L2 | DRD5 | DRD5_HUMAN | dopamine receptor D5
Type:
Protein
Mol. Mass.:
52943.41
Organism:
Homo sapiens (Human)
Description:
P21918
Residue:
477
Sequence:
MLPPGSNGTAYPGQFALYQQLAQGNAVGGSAGAPPLGPSQVVTACLLTLLIIWTLLGNVLVCAAIVRSRHLRANMTNVFIVSLAVSDLFVALLVMPWKAVAEVAGYWPFGAFCDVWVAFDIMCSTASILNLCVISVDRYWAISRPFRYKRKMTQRMALVMVGLAWTLSILISFIPVQLNWHRDQAASWGGLDLPNNLANWTPWEEDFWEPDVNAENCDSSLNRTYAISSSLISFYIPVAIMIVTYTRIYRIAQVQIRRISSLERAAEHAQSCRSSAACAPDTSLRASIKKETKVLKTLSVIMGVFVCCWLPFFILNCMVPFCSGHPEGPPAGFPCVSETTFDVFVWFGWANSSLNPVIYAFNADFQKVFAQLLGCSHFCSRTPVETVNISNELISYNQDIVFHKEIAAAYIHMMPNAVTPGNREVDNDEEEGPFDRMFQIYQTSPDGDPVAESVWELDCEGEISLDKITPFTPNGFH
  
Inhibitor
Name:
BDBM48967
Synonyms:
MLS000116741 | N-(2-oxolanylmethyl)-4-tetrazolo[1,5-a]quinoxalinamine | N-(oxolan-2-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]quinoxalin-4-amine | N-(oxolan-2-ylmethyl)tetrazolo[1,5-a]quinoxalin-4-amine | SMR000093700 | cid_5307548 | tetrahydrofurfuryl(tetrazolo[1,5-a]quinoxalin-4-yl)amine
Type:
Small organic molecule
Emp. Form.:
C13H14N6O
Mol. Mass.:
270.2899
SMILES:
C(Nc1nc2ccccc2n2nnnc12)C1CCCO1
Structure:
Search PDB for entries with ligand similarity: