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Target
DNA repair protein RAD51 homolog 1
Ligand
BDBM51360
Substrate
n/a
Meas. Tech.
Homologous recombination_Rad 51_dose response_2
IC50
53000±n/a nM
Citation
 PubChem, PC Homologous recombination_Rad 51_dose response_2 PubChem Bioassay (2008)[AID] 
Target
Name:
DNA repair protein RAD51 homolog 1
Synonyms:
RAD51 | RAD51A | RAD51_HUMAN | RECA
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36960.74
Organism:
Homo sapiens (Human)
Description:
gi_49168602
Residue:
339
Sequence:
MAMQMQLEANADTSVEEESFGPQPISRLEQCGINANDVKKLEEAGFHTVEAVAYAPKKELINIKGISEAKADKILAEAAKLVPMGFTTATEFHQRRSEIIQITTGSKELDKLLQGGIETGSITEMFGEFRTGKTQICHTLAVTCQLPIDRGGGEGKAMYIDTEGTFRPERLLAVAERYGLSGSDVLDNVAYARAFNTDHQTQLLYQASAMMVESRYALLIVDSATALYRTDYSGRGELSARQMHLARFLRMLLRLADEFGVAVVITNQVVAQVDGAAMFAADPKKPIGGNIIAHASTTRLYLRKGRGETRICKIYDSPCLPEAEAMFAINADGVGDAKD
  
Inhibitor
Name:
BDBM51360
Synonyms:
5-chloranyl-1,3-dimethyl-N-[2-oxidanylidene-2-[(phenylmethyl)amino]ethyl]pyrazole-4-carboxamide | 5-chloro-1,3-dimethyl-N-[2-oxo-2-[(phenylmethyl)amino]ethyl]-4-pyrazolecarboxamide | MLS000763400 | N-[2-(benzylamino)-2-keto-ethyl]-5-chloro-1,3-dimethyl-pyrazole-4-carboxamide | N-[2-(benzylamino)-2-oxoethyl]-5-chloro-1,3-dimethyl-1H-pyrazole-4-carboxamide | N-[2-(benzylamino)-2-oxoethyl]-5-chloro-1,3-dimethylpyrazole-4-carboxamide | SMR000336268 | cid_4421157
Type:
Small organic molecule
Emp. Form.:
C15H17ClN4O2
Mol. Mass.:
320.774
SMILES:
Cc1nn(C)c(Cl)c1C(=O)NCC(=O)NCc1ccccc1
Structure:
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