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Target
Regulator of G-protein signaling 4
Ligand
BDBM47830
Substrate
n/a
Meas. Tech.
Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao.
EC50
30000±n/a nM
Citation
 PubChem, PC Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 4
Synonyms:
RGP4 | RGS4 | RGS4_HUMAN | Regulator of G-protein signaling 4 (RGS4)
Type:
Enzyme
Mol. Mass.:
23263.51
Organism:
Homo sapiens (Human)
Description:
P49798
Residue:
205
Sequence:
MCKGLAGLPASCLRSAKDMKHRLGFLLQKSDSCEHNSSHNKKDKVVICQRVSQEEVKKWAESLENLISHECGLAAFKAFLKSEYSEENIDFWISCEEYKKIKSPSKLSPKAKKIYNEFISVQATKEVNLDSCTREETSRNMLEPTITCFDEAQKKIFNLMEKDSYRRFLKSRFYLDLVNPSSCGAEKQKGAKSSADCASLVPQCA
  
Inhibitor
Name:
BDBM47830
Synonyms:
4-cyclopropyl-6-(methylthio)-1,3,5-triazin-2-amine | 4-cyclopropyl-6-methylsulfanyl-1,3,5-triazin-2-amine | MLS000861275 | SMR000460059 | [4-cyclopropyl-6-(methylthio)-s-triazin-2-yl]amine | cid_602660
Type:
Small organic molecule
Emp. Form.:
C7H10N4S
Mol. Mass.:
182.246
SMILES:
CSc1nc(N)nc(n1)C1CC1
Structure:
Search PDB for entries with ligand similarity: