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Target
POsterior Segregation
Ligand
BDBM52069
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
39204±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM52069
Synonyms:
MLS000074775 | SMR000006509 | [4-(5-Fluoro-benzotriazol-1-yl)-piperidin-1-yl]-morpholin-4-yl-methanone | [4-(5-fluoranylbenzotriazol-1-yl)piperidin-1-yl]-morpholin-4-yl-methanone | [4-(5-fluoro-1-benzotriazolyl)-1-piperidinyl]-(4-morpholinyl)methanone | [4-(5-fluorobenzotriazol-1-yl)piperidin-1-yl]-morpholin-4-ylmethanone | [4-(5-fluorobenzotriazol-1-yl)piperidino]-morpholino-methanone | cid_649399
Type:
Small organic molecule
Emp. Form.:
C16H20FN5O2
Mol. Mass.:
333.3607
SMILES:
Fc1ccc2n(nnc2c1)C1CCN(CC1)C(=O)N1CCOCC1
Structure:
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