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Target
Kallikrein-5
Ligand
BDBM32676
Substrate
n/a
Meas. Tech.
Kallikrein 5 1536 HTS Dose Response Confirmation
IC50
275.07±n/a nM
Citation
 PubChem, PC Kallikrein 5 1536 HTS Dose Response Confirmation PubChem Bioassay (2008)[AID] 
Target
Name:
Kallikrein-5
Synonyms:
KLK5 | KLK5_HUMAN | Kallikrein 5 | SCTE | kallikrein-related peptidase 5 preproprotein
Type:
PROTEIN
Mol. Mass.:
32031.72
Organism:
Homo sapiens (Human)
Description:
EBI_12584
Residue:
293
Sequence:
MATARPPWMWVLCALITALLLGVTEHVLANNDVSCDHPSNTVPSGSNQDLGAGAGEDARSDDSSSRIINGSDCDMHTQPWQAALLLRPNQLYCGAVLVHPQWLLTAAHCRKKVFRVRLGHYSLSPVYESGQQMFQGVKSIPHPGYSHPGHSNDLMLIKLNRRIRPTKDVRPINVSSHCPSAGTKCLVSGWGTTKSPQVHFPKVLQCLNISVLSQKRCEDAYPRQIDDTMFCAGDKAGRDSCQGDSGGPVVCNGSLQGLVSWGDYPCARPNRPGVYTNLCKFTKWIQETIQANS
  
Inhibitor
Name:
BDBM32676
Synonyms:
(3-amino-1,2,4-triazol-4-yl)-(3,5-dimethylphenyl)methanone | (3-azanyl-1,2,4-triazol-4-yl)-(3,5-dimethylphenyl)methanone | 4-(3,5-dimethylbenzoyl)-4H-1,2,4-triazol-3-amine | MLS000063609 | SMR000075231 | cid_912604
Type:
Small organic molecule
Emp. Form.:
C11H12N4O
Mol. Mass.:
216.2392
SMILES:
Cc1cc(C)cc(c1)C(=O)n1cnnc1N
Structure:
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