Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 1
Ligand
BDBM61824
Substrate
n/a
Meas. Tech.
Fluorescence-based counterscreen for agonists of NPY-Y2: cell-based high-throughput dose response assay for agonists of NPY-Y1.
EC50
9924±n/a nM
Citation
 PubChem, PC Fluorescence-based counterscreen for agonists of NPY-Y2: cell-based high-throughput dose response assay for agonists of NPY-Y1. PubChem Bioassay (2009)[AID] 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44399.07
Organism:
Homo sapiens (Human)
Description:
NPY-Y1 NPY1R HUMAN::P25929
Residue:
384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
  
Inhibitor
Name:
BDBM61824
Synonyms:
2-[(2-methyl-5-oxidanylidene-3-phenyl-4H-imidazol-4-yl)diazenyl]benzoic acid | 2-[(2-methyl-5-oxo-3-phenyl-4H-imidazol-4-yl)azo]benzoic acid | 2-[(2-methyl-5-oxo-3-phenyl-4H-imidazol-4-yl)diazenyl]benzoic acid | 2-[(5-keto-2-methyl-3-phenyl-2-imidazolin-4-yl)azo]benzoic acid | MLS000713819 | SMR000273300 | cid_3117655
Type:
Small organic molecule
Emp. Form.:
C17H14N4O3
Mol. Mass.:
322.3181
SMILES:
Cc1nc(O)c(N=Nc2ccccc2C(O)=O)n1-c1ccccc1 |w:6.5|
Structure:
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