Target
Neuropeptides B/W receptor type 1
Ligand
BDBM62131
Substrate
n/a
Meas. Tech.
Fluorescence-based dose response cell-based high throughput screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7).
IC50
6654±n/a nM
Citation
 PubChem, PC Fluorescence-based dose response cell-based high throughput screening assay to identify antagonists of the G-protein coupled receptor 7 (GPR7). PubChem Bioassay (2010)[AID] 
Target
Name:
Neuropeptides B/W receptor type 1
Synonyms:
GPR7 | NPBW1_HUMAN | NPBWR1 | neuropeptides B/W receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36111.82
Organism:
Homo sapiens (Human)
Description:
gi_119607128
Residue:
328
Sequence:
MDNASFSEPWPANASGPDPALSCSNASTLAPLPAPLAVAVPVVYAVICAVGLAGNSAVLYVLLRAPRMKTVTNLFILNLAIADELFTLVLPINIADFLLRQWPFGELMCKLIVAIDQYNTFSSLYFLTVMSADRYLVVLATAESRRVAGRTYSAARAVSLAVWGIVTLVVLPFAVFARLDDEQGRRQCVLVFPQPEAFWWRASRLYTLVLGFAIPVSTICVLYTTLLCRLHAMRLDSHAKALERAKKRVTFLVVAILAVCLLCWTPYHLSTVVALTTDLPQTPLVIAISYFITSLSYANSCLNPFLYAFLDASFRRNLRQLITCRAAA
  
Inhibitor
Name:
BDBM62131
Synonyms:
MLS000974462 | N-[(2,3-dimethylanilino)-sulfanylidenemethyl]-2-phenylacetamide | N-[(2,3-dimethylphenyl)carbamothioyl]-2-phenyl-ethanamide | N-[(2,3-dimethylphenyl)carbamothioyl]-2-phenylacetamide | N-[(2,3-dimethylphenyl)thiocarbamoyl]-2-phenyl-acetamide | N-{[(2,3-dimethylphenyl)amino]carbonothioyl}-2-phenylacetamide | SMR000497992 | cid_952248
Type:
Small organic molecule
Emp. Form.:
C17H18N2OS
Mol. Mass.:
298.403
SMILES:
Cc1cccc(NC(=S)NC(=O)Cc2ccccc2)c1C
Structure:
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