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Target
Trans-activator protein BZLF1
Ligand
BDBM62411
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62411
Synonyms:
2-(2-Cyano-phenoxy)-N-(2-cyclopropanecarbonyl-benzofuran-3-yl)-acetamide | 2-(2-cyanophenoxy)-N-(2-cyclopropylcarbonyl-1-benzofuran-3-yl)ethanamide | 2-(2-cyanophenoxy)-N-[2-(cyclopropanecarbonyl)-1-benzofuran-3-yl]acetamide | 2-(2-cyanophenoxy)-N-[2-(cyclopropanecarbonyl)benzofuran-3-yl]acetamide | 2-(2-cyanophenoxy)-N-[2-[cyclopropyl(oxo)methyl]-3-benzofuranyl]acetamide | MLS000033658 | SMR000014220 | cid_654231
Type:
Small organic molecule
Emp. Form.:
C21H16N2O4
Mol. Mass.:
360.3627
SMILES:
O=C(COc1ccccc1C#N)Nc1c(oc2ccccc12)C(=O)C1CC1
Structure:
Search PDB for entries with ligand similarity: