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Target
Trans-activator protein BZLF1
Ligand
BDBM56866
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM56866
Synonyms:
MLS000531165 | N-[4-(2,6-dimethylpiperidin-1-yl)sulfonylphenyl]-3-(4-oxidanylidenequinazolin-3-yl)propanamide | N-[4-(2,6-dimethylpiperidin-1-yl)sulfonylphenyl]-3-(4-oxoquinazolin-3-yl)propanamide | N-[4-(2,6-dimethylpiperidino)sulfonylphenyl]-3-(4-ketoquinazolin-3-yl)propionamide | N-[4-[(2,6-dimethyl-1-piperidinyl)sulfonyl]phenyl]-3-(4-oxo-3-quinazolinyl)propanamide | N-{4-[(2,6-dimethyl-1-piperidinyl)sulfonyl]phenyl}-3-(4-oxo-3(4H)-quinazolinyl)propanamide | SMR000136143 | cid_2964209
Type:
Small organic molecule
Emp. Form.:
C24H28N4O4S
Mol. Mass.:
468.569
SMILES:
CC1CCCC(C)N1S(=O)(=O)c1ccc(NC(=O)CCn2cnc3ccccc3c2=O)cc1
Structure:
Search PDB for entries with ligand similarity: