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Target
Trans-activator protein BZLF1
Ligand
BDBM62444
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62444
Synonyms:
2-{N'-[5-(Benzenesulfonylamino-methyl)-furan-2-ylmethylene]-hydrazino}-N-(4-ethoxy-phenyl)-2-oxo-acetamide | MLS000554619 | N'-[[5-(benzenesulfonamidomethyl)-2-furanyl]methylideneamino]-N-(4-ethoxyphenyl)oxamide | N'-[[5-(benzenesulfonamidomethyl)-2-furyl]methyleneamino]-N-p-phenetyl-oxamide | N'-[[5-(benzenesulfonamidomethyl)furan-2-yl]methylideneamino]-N-(4-ethoxyphenyl)oxamide | N-(4-ethoxyphenyl)-N'-[[5-(phenylsulfonylaminomethyl)furan-2-yl]methylideneamino]ethanediamide | SMR000172100 | cid_3139240
Type:
Small organic molecule
Emp. Form.:
C22H22N4O6S
Mol. Mass.:
470.498
SMILES:
CCOc1ccc(NC(=O)C(=O)NN=Cc2ccc(CNS(=O)(=O)c3ccccc3)o2)cc1
Structure:
Search PDB for entries with ligand similarity: