Target
Trans-activator protein BZLF1
Ligand
BDBM62446
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62446
Synonyms:
MLS000560410 | N-(2-Phenylcarbamoylmethylsulfanyl-benzothiazol-6-yl)-2-(1-phenyl-1H-tetrazol-5-ylsulfanyl)-acetamide | N-[2-(2-anilino-2-oxoethyl)sulfanyl-1,3-benzothiazol-6-yl]-2-(1-phenyltetrazol-5-yl)sulfanylacetamide | N-[2-(2-oxidanylidene-2-phenylazanyl-ethyl)sulfanyl-1,3-benzothiazol-6-yl]-2-[(1-phenyl-1,2,3,4-tetrazol-5-yl)sulfanyl]ethanamide | N-[2-[(2-anilino-2-keto-ethyl)thio]-1,3-benzothiazol-6-yl]-2-[(1-phenyltetrazol-5-yl)thio]acetamide | N-[2-[(2-anilino-2-oxoethyl)thio]-1,3-benzothiazol-6-yl]-2-[(1-phenyl-5-tetrazolyl)thio]acetamide | SMR000176894 | cid_3130874
Type:
Small organic molecule
Emp. Form.:
C24H19N7O2S3
Mol. Mass.:
533.648
SMILES:
O=C(CSc1nc2ccc(NC(=O)CSc3nnnn3-c3ccccc3)cc2s1)Nc1ccccc1
Structure:
Search PDB for entries with ligand similarity: