Target
Trans-activator protein BZLF1
Ligand
BDBM62449
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62449
Synonyms:
(E)-2-cyano-3-[1-(2-fluorobenzyl)indol-3-yl]-N-(2-furfuryl)acrylamide | (E)-2-cyano-3-[1-[(2-fluorophenyl)methyl]-3-indolyl]-N-(2-furanylmethyl)-2-propenamide | (E)-2-cyano-3-[1-[(2-fluorophenyl)methyl]indol-3-yl]-N-(furan-2-ylmethyl)prop-2-enamide | 2-Cyano-3-[1-(2-fluoro-benzyl)-1H-indol-3-yl]-N-furan-2-ylmethyl-acrylamide | MLS000567542 | SMR000177355 | cid_1073562
Type:
Small organic molecule
Emp. Form.:
C24H18FN3O2
Mol. Mass.:
399.417
SMILES:
Fc1ccccc1Cn1cc(\C=C(/C#N)C(=O)NCc2ccco2)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: