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Target
Trans-activator protein BZLF1
Ligand
BDBM62454
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62454
Synonyms:
2-[6-(1,3-benzodioxol-5-yl)pyridazin-3-yl]sulfanyl-N-(3-fluoranyl-4-methyl-phenyl)ethanamide | 2-[6-(1,3-benzodioxol-5-yl)pyridazin-3-yl]sulfanyl-N-(3-fluoro-4-methylphenyl)acetamide | 2-[[6-(1,3-benzodioxol-5-yl)-3-pyridazinyl]thio]-N-(3-fluoro-4-methylphenyl)acetamide | 2-[[6-(1,3-benzodioxol-5-yl)pyridazin-3-yl]thio]-N-(3-fluoro-4-methyl-phenyl)acetamide | MLS000724890 | SMR000237115 | cid_7206330
Type:
Small organic molecule
Emp. Form.:
C20H16FN3O3S
Mol. Mass.:
397.423
SMILES:
Cc1ccc(NC(=O)CSc2ccc(nn2)-c2ccc3OCOc3c2)cc1F
Structure:
Search PDB for entries with ligand similarity: