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Target
Trans-activator protein BZLF1
Ligand
BDBM57703
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM57703
Synonyms:
MLS000394802 | N-[(Z)-(1-methyl-2-oxidanylidene-indol-3-ylidene)amino]-2-thiophen-2-yl-quinoline-4-carboxamide | N-[(Z)-(1-methyl-2-oxo-3-indolylidene)amino]-2-thiophen-2-yl-4-quinolinecarboxamide | N-[(Z)-(1-methyl-2-oxoindol-3-ylidene)amino]-2-thiophen-2-ylquinoline-4-carboxamide | N-[(Z)-(2-keto-1-methyl-indolin-3-ylidene)amino]-2-(2-thienyl)cinchoninamide | SMR000242891 | cid_6901801
Type:
Small organic molecule
Emp. Form.:
C23H16N4O2S
Mol. Mass.:
412.464
SMILES:
CN1C(=O)\C(=N/NC(=O)c2cc(nc3ccccc23)-c2cccs2)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: