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Target
Trans-activator protein BZLF1
Ligand
BDBM61180
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM61180
Synonyms:
MLS000528436 | N-[4-(2-{[(Furan-2-ylmethyl)-carbamoyl]-methyl}-2H-tetrazol-5-yl)-phenyl]-2-methoxy-benzamide | N-[4-[2-[2-(2-furanylmethylamino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-methoxybenzamide | N-[4-[2-[2-(2-furfurylamino)-2-keto-ethyl]tetrazol-5-yl]phenyl]-2-methoxy-benzamide | N-[4-[2-[2-(furan-2-ylmethylamino)-2-oxidanylidene-ethyl]-1,2,3,4-tetrazol-5-yl]phenyl]-2-methoxy-benzamide | N-[4-[2-[2-(furan-2-ylmethylamino)-2-oxoethyl]tetrazol-5-yl]phenyl]-2-methoxybenzamide | SMR000121011 | cid_1452563
Type:
Small organic molecule
Emp. Form.:
C22H20N6O4
Mol. Mass.:
432.432
SMILES:
COc1ccccc1C(=O)Nc1ccc(cc1)-c1nnn(CC(=O)NCc2ccco2)n1
Structure:
Search PDB for entries with ligand similarity: