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Target
Trans-activator protein BZLF1
Ligand
BDBM34345
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM34345
Synonyms:
2-[2-(5-morpholin-4-ylsulfonylthiophen-2-yl)ethanoylamino]-5-phenyl-thiophene-3-carboxamide | 2-[[2-(5-morpholin-4-ylsulfonylthiophen-2-yl)acetyl]amino]-5-phenylthiophene-3-carboxamide | 2-[[2-(5-morpholinosulfonyl-2-thienyl)acetyl]amino]-5-phenyl-thiophene-3-carboxamide | 2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamide | MLS000053467 | SMR000063575 | cid_2121076
Type:
Small organic molecule
Emp. Form.:
C21H21N3O5S3
Mol. Mass.:
491.604
SMILES:
NC(=O)c1cc(sc1NC(=O)Cc1ccc(s1)S(=O)(=O)N1CCOCC1)-c1ccccc1
Structure:
Search PDB for entries with ligand similarity: