Target
Trans-activator protein BZLF1
Ligand
BDBM62497
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62497
Synonyms:
4-[2-[[2-(4-methyl-1-piperidinyl)-1-oxoethyl]amino]-4-thiazolyl]benzoic acid ethyl ester | 4-[2-[[2-(4-methylpiperidino)acetyl]amino]thiazol-4-yl]benzoic acid ethyl ester | MLS001175133 | SMR000595579 | cid_2334129 | ethyl 4-[2-[2-(4-methylpiperidin-1-yl)ethanoylamino]-1,3-thiazol-4-yl]benzoate | ethyl 4-[2-[[2-(4-methylpiperidin-1-yl)acetyl]amino]-1,3-thiazol-4-yl]benzoate
Type:
Small organic molecule
Emp. Form.:
C20H25N3O3S
Mol. Mass.:
387.496
SMILES:
CCOC(=O)c1ccc(cc1)-c1csc(NC(=O)CN2CCC(C)CC2)n1
Structure:
Search PDB for entries with ligand similarity: