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Target
Trans-activator protein BZLF1
Ligand
BDBM62516
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62516
Synonyms:
5-methoxy-3-methyl-2-benzofurancarboxylic acid [2-[2-methyl-5-(4-morpholinylsulfonyl)anilino]-2-oxoethyl] ester | 5-methoxy-3-methyl-coumarilic acid [2-keto-2-(2-methyl-5-morpholinosulfonyl-anilino)ethyl] ester | MLS001099519 | SMR000715706 | [2-(2-methyl-5-morpholin-4-ylsulfonylanilino)-2-oxoethyl] 5-methoxy-3-methyl-1-benzofuran-2-carboxylate | [2-[(2-methyl-5-morpholin-4-ylsulfonyl-phenyl)amino]-2-oxidanylidene-ethyl] 5-methoxy-3-methyl-1-benzofuran-2-carboxylate | cid_24687714
Type:
Small organic molecule
Emp. Form.:
C24H26N2O8S
Mol. Mass.:
502.537
SMILES:
COc1ccc2oc(C(=O)OCC(=O)Nc3cc(ccc3C)S(=O)(=O)N3CCOCC3)c(C)c2c1
Structure:
Search PDB for entries with ligand similarity: