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Target
Mu-type opioid receptor
Ligand
BDBM64847
Substrate
n/a
Meas. Tech.
Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1)
IC50
5107±n/a nM
Citation
 PubChem, PC Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay (2010)[AID] 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Homo sapiens (Human)
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM64847
Synonyms:
3-Chloro-6-methoxy-benzo[b]thiophene-2-carboxylic acid benzo[1,3]dioxol-5-ylmethylene-hydrazide | 3-chloro-6-methoxy-N-(piperonylideneamino)benzothiophene-2-carboxamide | MLS000549759 | N-(1,3-benzodioxol-5-ylmethylideneamino)-3-chloranyl-6-methoxy-1-benzothiophene-2-carboxamide | N-(1,3-benzodioxol-5-ylmethylideneamino)-3-chloro-6-methoxy-1-benzothiophene-2-carboxamide | SMR000175212 | cid_1369102
Type:
Small organic molecule
Emp. Form.:
C18H13ClN2O4S
Mol. Mass.:
388.825
SMILES:
COc1ccc2c(Cl)c(sc2c1)C(=O)NN=Cc1ccc2OCOc2c1
Structure:
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