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Target
Mu-type opioid receptor
Ligand
BDBM64868
Substrate
n/a
Meas. Tech.
Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1)
IC50
5818±n/a nM
Citation
 PubChem, PC Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay (2010)[AID] 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Homo sapiens (Human)
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM64868
Synonyms:
5-(3,4-dichlorophenyl)-1-phenyl-1H-pyrazole-3-carboxylic acid | 5-(3,4-dichlorophenyl)-1-phenyl-3-pyrazolecarboxylic acid | 5-(3,4-dichlorophenyl)-1-phenyl-pyrazole-3-carboxylic acid | 5-(3,4-dichlorophenyl)-1-phenylpyrazole-3-carboxylic acid | MLS001166361 | SMR000549909 | cid_1477263
Type:
Small organic molecule
Emp. Form.:
C16H10Cl2N2O2
Mol. Mass.:
333.169
SMILES:
OC(=O)c1cc(-c2ccc(Cl)c(Cl)c2)n(n1)-c1ccccc1
Structure:
Search PDB for entries with ligand similarity: