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Target
Trans-activator protein BZLF1
Ligand
BDBM64839
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64839
Synonyms:
2-(3,5-dimethyl-1-pyrazolyl)-4-(2-phenylethylamino)-5-pyrimidinecarboxylic acid ethyl ester | 2-(3,5-dimethylpyrazol-1-yl)-4-(phenethylamino)pyrimidine-5-carboxylic acid ethyl ester | MLS000040645 | SMR000043873 | cid_663159 | ethyl 2-(3,5-dimethylpyrazol-1-yl)-4-(2-phenylethylamino)pyrimidine-5-carboxylate
Type:
Small organic molecule
Emp. Form.:
C20H23N5O2
Mol. Mass.:
365.4289
SMILES:
CCOC(=O)c1cnc(nc1NCCc1ccccc1)-n1nc(C)cc1C
Structure:
Search PDB for entries with ligand similarity: