Target
Trans-activator protein BZLF1
Ligand
BDBM64852
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
45082±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64852
Synonyms:
5-methyl-N-(4-methylphenyl)-2-(2-pyridinyl)-3-imidazo[1,2-a]pyridinamine | 5-methyl-N-(4-methylphenyl)-2-pyridin-2-yl-imidazo[1,2-a]pyridin-3-amine | 5-methyl-N-(4-methylphenyl)-2-pyridin-2-ylimidazo[1,2-a]pyridin-3-amine | MLS000730306 | SMR000308582 | [5-methyl-2-(2-pyridyl)imidazo[1,2-a]pyridin-3-yl]-(p-tolyl)amine | cid_7066845
Type:
Small organic molecule
Emp. Form.:
C20H18N4
Mol. Mass.:
314.3837
SMILES:
Cc1ccc(Nc2c(nc3cccc(C)n23)-c2ccccn2)cc1
Structure:
Search PDB for entries with ligand similarity: