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Target
Trans-activator protein BZLF1
Ligand
BDBM64857
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64857
Synonyms:
5-methoxy-4-(4-methylphenyl)sulfanyl-2-pyridin-2-yl-pyrimidine | 5-methoxy-4-(4-methylphenyl)sulfanyl-2-pyridin-2-ylpyrimidine | 5-methoxy-4-(p-tolylthio)-2-(2-pyridyl)pyrimidine | 5-methoxy-4-[(4-methylphenyl)thio]-2-(2-pyridinyl)pyrimidine | MLS000692232 | SMR000333903 | cid_1470825 | methyl 4-[(4-methylphenyl)sulfanyl]-2-(2-pyridinyl)-5-pyrimidinyl ether
Type:
Small organic molecule
Emp. Form.:
C17H15N3OS
Mol. Mass.:
309.386
SMILES:
COc1cnc(nc1Sc1ccc(C)cc1)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: