Reaction Details Report a problem with these data
Target
Trans-activator protein BZLF1
Ligand
BDBM64867
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64867
Synonyms:
5-methoxy-2-(2-pyridinyl)-4-[3-(trifluoromethyl)phenoxy]pyrimidine | 5-methoxy-2-(2-pyridinyl)-4-pyrimidinyl 3-(trifluoromethyl)phenyl ether | 5-methoxy-2-(2-pyridyl)-4-[3-(trifluoromethyl)phenoxy]pyrimidine | 5-methoxy-2-pyridin-2-yl-4-[3-(trifluoromethyl)phenoxy]pyrimidine | MLS001165473 | SMR000549594 | cid_3792008
Type:
Small organic molecule
Emp. Form.:
C17H12F3N3O2
Mol. Mass.:
347.2913
SMILES:
COc1cnc(nc1Oc1cccc(c1)C(F)(F)F)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: