Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM67117
Substrate
n/a
Meas. Tech.
Late stage counterscreen results from the probe development effort to identify STAT1 inhibitors: luminescence-based cell-based dose response assay for STAT3 inhibitors
IC50
>55690±n/a nM
Citation
 PubChem, PC Late stage counterscreen results from the probe development effort to identify STAT1 inhibitors: luminescence-based cell-based dose response assay for STAT3 inhibitors PubChem Bioassay (2010)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM67117
Synonyms:
2-(4-besylpiperazino)-N-phenyl-propionamide | 2-[4-(benzenesulfonyl)-1-piperazinyl]-N-phenylpropanamide | 2-[4-(benzenesulfonyl)piperazin-1-yl]-N-phenylpropanamide | N-phenyl-2-[4-(phenylsulfonyl)piperazin-1-yl]propanamide | SR-03000000786-1 | cid_17453313
Type:
Small organic molecule
Emp. Form.:
C19H23N3O3S
Mol. Mass.:
373.469
SMILES:
CC(N1CCN(CC1)S(=O)(=O)c1ccccc1)C(=O)Nc1ccccc1
Structure:
Search PDB for entries with ligand similarity: