Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM51019
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
10093±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM51019
Synonyms:
4-methyl-7-benzo[a]phenalenone | 4-methyl-7H-benzo[de]anthracen-7-one | 4-methylbenzo[a]phenalen-7-one | MLS000585787 | SMR000204350 | cid_232704
Type:
Small organic molecule
Emp. Form.:
C18H12O
Mol. Mass.:
244.2873
SMILES:
Cc1ccc2C(=O)c3ccccc3-c3cccc1c23
Structure:
Search PDB for entries with ligand similarity: