Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67430
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
>75403±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67430
Synonyms:
2-methyl-5-[(4-methylphenyl)sulfonylamino]-N-phenyl-3-benzo[g]benzofurancarboxamide | 2-methyl-5-[(4-methylphenyl)sulfonylamino]-N-phenyl-benzo[g][1]benzofuran-3-carboxamide | 2-methyl-5-[(4-methylphenyl)sulfonylamino]-N-phenylbenzo[g][1]benzofuran-3-carboxamide | 2-methyl-N-phenyl-5-(tosylamino)benzo[g]benzofuran-3-carboxamide | MLS000394360 | SMR000248371 | cid_2337760
Type:
Small organic molecule
Emp. Form.:
C27H22N2O4S
Mol. Mass.:
470.54
SMILES:
Cc1oc2c(cc(NS(=O)(=O)c3ccc(C)cc3)c3ccccc23)c1C(=O)Nc1ccccc1
Structure:
Search PDB for entries with ligand similarity: