Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67432
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
>75487±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67432
Synonyms:
3-(trifluoromethyl)-1H-benzo[g]quinoxalin-2-one | 3-(trifluoromethyl)benzo[g]quinoxalin-2-ol | MLS000686612 | SMR000315133 | cid_1502798
Type:
Small organic molecule
Emp. Form.:
C13H7F3N2O
Mol. Mass.:
264.2027
SMILES:
FC(F)(F)c1nc2cc3ccccc3cc2[nH]c1=O
Structure:
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