Target
Protein Rev
Ligand
BDBM67445
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
22020±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67445
Synonyms:
2-(4-Hydroxyphenylazo)benzoic acid | 2-[2-(4-oxidanylidenecyclohexa-2,5-dien-1-ylidene)hydrazinyl]benzoic acid | 2-[2-(4-oxo-1-cyclohexa-2,5-dienylidene)hydrazinyl]benzoic acid | 2-[2-(4-oxocyclohexa-2,5-dien-1-ylidene)hydrazinyl]benzoic acid | 2-[N'-(4-ketocyclohexa-2,5-dien-1-ylidene)hydrazino]benzoic acid | MLS001174930 | SMR000471883 | cid_5357439
Type:
Small organic molecule
Emp. Form.:
C13H10N2O3
Mol. Mass.:
242.2301
SMILES:
OC(=O)c1ccccc1N=Nc1ccc(O)cc1 |w:9.9|
Structure:
Search PDB for entries with ligand similarity: