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Target
X-box-binding protein 1
Ligand
BDBM39089
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
210±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM39089
Synonyms:
2-(5-bromanyl-2-chloranyl-phenyl)-1,3-benzoxazol-5-amine | 2-(5-bromo-2-chlorophenyl)-1,3-benzoxazol-5-amine | MLS000036810 | SMR000036737 | [2-(5-bromo-2-chloro-phenyl)-1,3-benzoxazol-5-yl]amine | cid_659499
Type:
Small organic molecule
Emp. Form.:
C13H8BrClN2O
Mol. Mass.:
323.572
SMILES:
Nc1ccc2oc(nc2c1)-c1cc(Br)ccc1Cl
Structure:
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